The Athlete's Formulary
TAF
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TAF is intended solely for qualified healthcare professionals. It is a medication governance reference and does not provide diagnostic guidance. All clinical decisions, laboratory assessment, and final choice of agent remain the responsibility of the treating clinician. Anti-doping status must be independently verified via wada-ama.org or globaldro.com before any clinical decision with anti-doping implications. Full terms at Terms of Access.
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TAF
The Athlete's Formulary
Medication governance reference for sport
Beta — Restricted Access
HomeMedicinesAntibacterials

Antibacterials

TAF covers athlete-specific governance considerations for antibiotic use in elite sport. Indications, standard dosing, and contraindications are not covered here — refer to the BNF and individual SmPCs. Local sensitivity data should inform antibiotic prescribing decisions. Governance flag
Evidence Ratings: A Systematic review / meta-analysis of RCTs   B Individual RCT or strong observational data   C Cohort / mechanistic human studies   D Case series / preclinical / operational   E In vitro / theoretical
Cephalosporins
Class Profiles
Comparative Table
Cephalosporins — Class Overview
Cefalexin · Cefaclor · Cefuroxime axetil
WADA: Not Prohibited 2026
1 — Athlete-Specific Considerations

Cross-reactivity with penicillins is side-chain dependent rather than class-wide. Risk varies by agent based on R1 side-chain similarity to the culprit penicillin — see individual agent notes. A1

Antibiotic-associated diarrhoea (AAD): A class effect for cephalosporins, with risk varying by agent. Cefuroxime shown to be associated with a particularly elevated C. difficile-associated diarrhoea risk. B2 GI side effects may affect training nutrition and hydration around competition. See Field 4.

Microbiome impact: Varies by agent within this class — see individual agent notes. Probiotic consideration may be appropriate — see TAF Probiotics entry.

2 — Formulation and Route

Form: Oral tablets and capsules (cefalexin, cefaclor). Oral tablets (cefuroxime axetil).

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status of prescribed agent before international travel. Carry prescribing documentation when transporting medicines across borders.

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food interactions: Vary by agent. Cefuroxime axetil absorption significantly enhanced when taken with or shortly after food. See individual agent notes.

4 — Performance-Impact Risks

Antibiotic-associated diarrhoea (AAD): Cephalosporins carry a class-level AAD risk with variation by agent. AAD may affect hydration, electrolyte balance, and training nutrition during a course of treatment. Risk is higher with cefuroxime than with cefalexin or cefaclor. B2

GI side effects: Nausea, vomiting, and abdominal discomfort reported across the class. May affect dietary intake and training tolerance during treatment course.

Fatigue: Underlying infection rather than the antibiotic is the primary driver of fatigue and reduced performance capacity during treatment. TAF does not provide return-to-training guidance — this remains a clinical decision.

Photosensitivity: Not a significant concern for this class. No specific training or outdoor competition restrictions required on photosensitivity grounds.

5 — Recovery-Impact Risks

GI tolerability and training load: AAD and GI side effects during a cephalosporin course may affect an athlete's ability to maintain training nutrition and hydration targets, with downstream impact on recovery capacity.

Microbiome disruption: All three agents associated with gut flora changes to varying degrees — see individual agent notes. Microbiome disruption may affect recovery through altered nutrient absorption and gut barrier function. Probiotic consideration may be appropriate — see TAF Probiotics entry.

Sleep and fatigue: No direct evidence of cephalosporin-specific effects on sleep or recovery beyond those attributable to the underlying infection.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see individual agent SmPC for full interaction profile.

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Iron, calcium, magnesium, zinc: No clinically significant absorption interaction established for cephalosporins.

Proton pump inhibitors: Concurrent PPI use associated with increased CDAD risk in hospitalised populations. B2 Relevance in otherwise healthy athletes is lower but worth noting where PPIs are co-prescribed.

Oral contraceptives: No clinically significant interaction established for cephalosporins with combined oral contraceptives based on current evidence.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

All three agents are generic oral antibiotics available at low cost through NHS dispensing and private prescription. Indicative costs per unit in individual agent notes.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer and dispensed product. Verify per dispensed product SmPC.

Penicillin allergy: See Field 1 and individual agent notes for cross-reactivity risk by agent.

Lactose: Present in some tablet formulations. Verify per dispensed product.

Gelatin: Present in some capsule formulations. Not suitable for vegetarians, vegans, or those observing halal or kosher dietary requirements where gelatin is derived from non-compliant sources. Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

INDIVIDUAL AGENTS

Cefalexin
1st generation · Capsules and tablets · POM
POM Rx
1 — Athlete-Specific Considerations

First-generation oral cephalosporin. Narrow spectrum relative to second-generation agents within this class.

Penicillin cross-reactivity: Aminocephalosporin — estimated cross-reactivity 16.45% in confirmed aminopenicillin allergy. A1

Microbiome impact: Low to moderate. D4

AAD risk: Moderate. Lower than cefuroxime within this class.

2 — Formulation and Route

Form: Capsules and tablets. Oral suspension available.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label.

SmPC: Cefalexin SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Can be taken with or without food. Taking with food is recommended to minimise GI side effects during training.

4 — Performance-Impact Risks

AAD risk: Moderate within class. Less strongly associated with C. difficile-associated diarrhoea than cefuroxime. B2

GI side effects: Nausea and diarrhoea reported. Taking with food reduces GI side effects and is recommended during training periods.

Photosensitivity: Not a concern with cefalexin. No outdoor training restrictions required.

5 — Recovery-Impact Risks

GI tolerability: Generally well tolerated. GI side effects during a course may affect training nutrition and hydration targets.

Microbiome disruption: Low to moderate. Short-course impact likely limited and reversible. Probiotic consideration may be appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Iron, calcium, magnesium, zinc: No clinically significant absorption interaction established for cefalexin.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.09 per 500mg capsule.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Cefaclor
2nd generation · Capsules and tablets · POM
POM Rx
1 — Athlete-Specific Considerations

Second-generation oral cephalosporin. Broader spectrum than cefalexin.

Penicillin cross-reactivity: Aminocephalosporin — estimated cross-reactivity 16.45% in confirmed aminopenicillin allergy. A1

Microbiome impact: Low to moderate. Minor, reversible anaerobic flora changes documented in volunteer data. Normalisation within one week of stopping treatment. C3

AAD risk: Moderate. Class effect applies. Direct evidence for cefaclor-specific AAD risk is limited — risk inferred from cephalosporin class data. C3

2 — Formulation and Route

Form: Capsules and tablets. Modified-release tablets and oral suspension available.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label.

SmPC: Cefaclor SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Can be taken with or without food. Taking with food recommended to minimise GI side effects during training.

4 — Performance-Impact Risks

AAD risk: Moderate. Class effect applies. GI side effects may affect hydration, electrolyte balance, and training nutrition during treatment course.

GI side effects: Nausea and diarrhoea reported. Taking with food reduces GI side effects and is recommended during training periods.

Photosensitivity: Not a concern with cefaclor. No outdoor training restrictions required.

5 — Recovery-Impact Risks

GI tolerability: Generally well tolerated. GI side effects during a course may affect training nutrition and hydration targets.

Microbiome disruption: Low to moderate. Short-course impact limited and reversible within one week of stopping treatment. Probiotic consideration may be appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Iron, calcium, magnesium, zinc: No clinically significant absorption interaction established for cefaclor.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.36 per 500mg capsule.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Cefuroxime Axetil
2nd generation · Tablets · POM
POM Rx
1 — Athlete-Specific Considerations

Second-generation oral cephalosporin. Broader spectrum than cefalexin and cefaclor within this class.

Penicillin cross-reactivity: Intermediate R1 side-chain similarity to penicillins. Estimated cross-reactivity 5.6% in confirmed penicillin allergy. Lower risk than aminocephalosporins but not negligible. A1

Microbiome impact: Moderate. More noticeable dysbiosis than cefalexin or cefaclor consistent with broader spectrum. C5

AAD risk: Moderate to high. Cefuroxime associated with significantly elevated C. difficile-associated diarrhoea risk. B2

2 — Formulation and Route

Form: Tablets.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label.

SmPC: Cefuroxime axetil SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Absorption significantly enhanced when taken with or shortly after food. Taking with food is recommended and improves bioavailability as well as reducing GI side effects during training.

4 — Performance-Impact Risks

AAD risk: Moderate to high. Cefuroxime associated with significantly elevated C. difficile-associated diarrhoea risk. May affect hydration, electrolyte balance, and training nutrition during treatment course. B2

GI side effects: Nausea and diarrhoea reported. Taking with food reduces GI side effects and is recommended during training periods.

Photosensitivity: Not a concern with cefuroxime axetil. No outdoor training restrictions required.

5 — Recovery-Impact Risks

GI tolerability: Higher GI risk within this class. AAD and GI side effects during a course may affect training nutrition and hydration targets more significantly than with cefalexin or cefaclor.

Microbiome disruption: Moderate. Broader spectrum associated with more noticeable dysbiosis than first-generation agents. Probiotic consideration may be appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Iron, calcium, magnesium, zinc: No clinically significant absorption interaction established for cefuroxime axetil.

Antacids and acid-suppressing medicines (PPIs, H2 antagonists): Medicines that reduce gastric acidity may reduce cefuroxime axetil bioavailability and cancel the absorption benefit of taking with food. SmPC Concurrent PPI use also associated with increased CDAD risk where cefuroxime is prescribed. B2

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.65 per 250mg tablet.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Fluoroquinolones
MHRA Safety Restriction — January 2024

Systemic fluoroquinolones must only be prescribed when other commonly recommended antibiotics are inappropriate. Situations where use may be appropriate include resistance to first-line antibiotics, contraindication to first-line antibiotics, side effects requiring cessation of first-line treatment, or failure of first-line treatment.

Tendon damage: Risk of tendinitis and tendon rupture. Onset may occur within 48 hours of starting treatment or be delayed for months after stopping. Risk significantly increased by concurrent corticosteroid use — a common combination in elite sport.

Disabling and potentially irreversible side effects affecting musculoskeletal, neurological, psychiatric and sensory systems have been reported. Estimated minimum frequency 1 in 10,000 patients.

Stop immediately and seek medical review at first signs of tendon pain or swelling, joint pain or swelling, abnormal sensations, muscle weakness, severe fatigue, mood disturbance, sleep disorder, or changes in vision, taste, smell or hearing.

Source: MHRA Drug Safety Update. January 2024. Full guidance ↗

Class Profiles
Comparative Table
Fluoroquinolones — Class Overview
Ciprofloxacin · Levofloxacin
WADA: Not Prohibited 2026
1 — Athlete-Specific Considerations

Fluoroquinolones are broad-spectrum antibiotics subject to MHRA prescribing restrictions since January 2024. See warning box above.

Tendon risk: Significantly elevated in athletes due to high training loads, concurrent corticosteroid use, and pre-existing tendon stress. Risk of tendinitis and tendon rupture applies to all tendons — Achilles tendon most commonly reported. See individual agent notes.

QTc prolongation: Class effect. In athletes where cardiac screening has not been undertaken, QTc-prolonging antibiotics warrant additional clinical consideration before prescribing.

CNS effects: Insomnia, anxiety, dizziness, and mood disturbance reported. Directly relevant to sleep quality, recovery, and performance during treatment course.

Photosensitivity: Significant class effect. Relevant for outdoor athletes — see individual agent notes and Field 3.

Microbiome impact: High. Significant dysbiosis reported with fluoroquinolone use, with some studies reporting effects persisting up to one year. Probiotic consideration appropriate — see TAF Probiotics entry.

AAD risk: High. See Field 4.

2 — Formulation and Route

Form: Oral tablets (ciprofloxacin, levofloxacin).

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel — fluoroquinolone availability and legal status varies by jurisdiction.

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Can be taken with or without food. Taking with food recommended to minimise GI side effects. Avoid taking with dairy products or calcium-fortified foods and drinks as these reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Supplement timing: Iron, calcium, magnesium, zinc, and multivitamin supplements taken at the same time as fluoroquinolones significantly reduce antibiotic absorption. Separate fluoroquinolone dosing from these supplements by at least two hours before or six hours after.

Outdoor training and photosensitivity: Avoid prolonged sun exposure during treatment course. Additional sun protection measures recommended for outdoor training and competition — see individual agent notes.

4 — Performance-Impact Risks

Tendon risk: Significantly elevated in athletes. Tendinitis and tendon rupture risk applies to all tendons. Achilles tendon most commonly reported. Concurrent corticosteroid use markedly increases risk. Stop treatment immediately at first signs of tendon pain or swelling and seek medical review.

CNS effects: Insomnia, anxiety, dizziness, and mood disturbance reported. May affect sleep quality, concentration, and performance during treatment course.

Photosensitivity: Significant class effect. Avoid prolonged sun exposure during treatment. Relevant for outdoor training and competition — sun protection measures required.

AAD risk: High. GI side effects including diarrhoea may affect hydration, electrolyte balance, and training nutrition during treatment course.

GI side effects: Nausea, vomiting, and abdominal discomfort reported. Taking with food recommended during training periods. Avoid dairy and calcium-fortified foods at time of dosing.

5 — Recovery-Impact Risks

Tendon and musculoskeletal: Tendon damage may present during or months after completing a course. Athletes returning to full training following fluoroquinolone use should be aware of delayed onset tendon symptoms. Clinical review warranted at first signs of tendon pain or swelling.

CNS and sleep: Insomnia and mood disturbance may affect recovery quality during treatment course. Sleep disruption compounds training load stress.

Microbiome disruption: High. Significant reduction in gut microbial diversity reported, with some evidence of effects persisting up to one year after stopping treatment. May affect nutrient absorption and gut barrier function. Probiotic consideration appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see individual agent SmPC for full interaction profile.

Iron, calcium, magnesium, zinc, and multivitamins: Significantly reduce fluoroquinolone absorption when taken concurrently. Separate dosing by at least two hours before or six hours after fluoroquinolone dose.

Dairy and calcium-fortified foods and drinks: Reduce fluoroquinolone absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Corticosteroids: Concurrent use significantly increases risk of tendinitis and tendon rupture. Avoid co-administration where possible. [MHRA 2024]

NSAIDs: Concurrent use may increase risk of CNS side effects including seizures. Caution warranted given prevalence of NSAID use in elite sport.

QTc-prolonging medicines: Additive QTc prolongation risk. Caution where athlete is prescribed other QTc-prolonging agents.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Generic oral antibiotics. Low cost through NHS dispensing and private prescription. Indicative costs per unit in individual agent notes.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

INDIVIDUAL AGENTS

Ciprofloxacin
Fluoroquinolone · Tablets · POM
POM Rx
1 — Athlete-Specific Considerations

Most widely prescribed fluoroquinolone in UK primary care. Broad-spectrum activity. Subject to MHRA 2024 prescribing restrictions — see class warning box.

Tendon risk: Applicable as per class. Achilles tendon most commonly reported. Risk increased with concurrent corticosteroid use, high training loads, and pre-existing tendon pathology.

Photosensitivity: Moderate. Relevant for outdoor athletes during treatment course.

QTc prolongation: Class effect. Lower QTc risk than moxifloxacin but not negligible. Relevant in athletes with unscreened cardiac status.

Microbiome impact: High. Significant reduction in gut microbial diversity reported, with some evidence of effects persisting up to one year after stopping treatment. C6

AAD risk: High.

2 — Formulation and Route

Form: Tablets.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Ciprofloxacin SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Can be taken with or without food. Taking with food recommended to minimise GI side effects. Avoid taking with dairy products or calcium-fortified foods and drinks as these reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Supplement timing: Iron, calcium, magnesium, zinc, and multivitamin supplements significantly reduce ciprofloxacin absorption. Separate dosing by at least two hours before or six hours after ciprofloxacin dose.

Outdoor training and photosensitivity: Avoid prolonged sun exposure during treatment course. Additional sun protection measures recommended for outdoor training and competition.

4 — Performance-Impact Risks

Tendon risk: Applicable as per class warning. Stop immediately at first signs of tendon pain or swelling.

CNS effects: Insomnia, anxiety, and dizziness reported. May affect sleep quality and performance during treatment course.

Photosensitivity: Moderate. Sun protection required for outdoor training and competition.

AAD risk: High. GI side effects may affect hydration, electrolyte balance, and training nutrition.

GI side effects: Nausea and diarrhoea reported. Taking with food recommended during training periods. Avoid dairy and calcium-fortified foods at time of dosing.

5 — Recovery-Impact Risks

Tendon and musculoskeletal: Delayed onset tendon symptoms possible months after completing a course. Clinical review warranted at first signs of tendon pain or swelling following recent ciprofloxacin use.

CNS and sleep: Insomnia and anxiety may affect recovery quality during treatment course.

Microbiome disruption: High. Significant gut microbial diversity reduction reported, with effects potentially persisting up to one year. Probiotic consideration appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

Iron, calcium, magnesium, zinc, and multivitamins: Significantly reduce ciprofloxacin absorption. Separate dosing by at least two hours before or six hours after ciprofloxacin dose.

Dairy and calcium-fortified foods and drinks: Reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Corticosteroids: Concurrent use significantly increases tendon rupture risk. Avoid co-administration where possible. [MHRA 2024]

NSAIDs: Concurrent use may increase risk of CNS side effects including seizures. Caution warranted given prevalence of NSAID use in elite sport.

Caffeine: Ciprofloxacin inhibits caffeine metabolism, increasing plasma caffeine levels. Athletes using caffeine as a performance supplement should be aware of potential for increased caffeine side effects during a ciprofloxacin course.

QTc-prolonging medicines: Additive QTc prolongation risk.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.39 per 500mg tablet.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Levofloxacin
Fluoroquinolone · Tablets · POM
POM Rx
1 — Athlete-Specific Considerations

Fluoroquinolone with activity broadly similar to ciprofloxacin but with enhanced gram-positive and atypical organism coverage. Subject to MHRA 2024 prescribing restrictions — see class warning box.

Tendon risk: Applicable as per class. Achilles tendon most commonly reported. Risk increased with concurrent corticosteroid use, high training loads, and pre-existing tendon pathology.

Photosensitivity: Moderate to high. More significant photosensitivity signal than ciprofloxacin. Relevant for outdoor athletes during treatment course.

QTc prolongation: Class effect. Higher QTc risk than ciprofloxacin. Relevant in athletes with unscreened cardiac status.

Microbiome impact: High. Significant reduction in gut microbial diversity reported. C6

AAD risk: High.

2 — Formulation and Route

Form: Tablets.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Levofloxacin SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Can be taken with or without food. Taking with food recommended to minimise GI side effects. Avoid taking with dairy products or calcium-fortified foods and drinks as these reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Supplement timing: Iron, calcium, magnesium, zinc, and multivitamin supplements significantly reduce levofloxacin absorption. Separate dosing by at least two hours before or six hours after levofloxacin dose.

Outdoor training and photosensitivity: Avoid prolonged sun exposure during treatment course. Additional sun protection measures recommended for outdoor training and competition. Photosensitivity risk higher than ciprofloxacin.

4 — Performance-Impact Risks

Tendon risk: Applicable as per class warning. Stop immediately at first signs of tendon pain or swelling.

CNS effects: Insomnia, anxiety, and dizziness reported. May affect sleep quality and performance during treatment course.

Photosensitivity: Moderate to high. More significant than ciprofloxacin. Sun protection required for all outdoor training and competition during treatment course.

AAD risk: High. GI side effects may affect hydration, electrolyte balance, and training nutrition.

GI side effects: Nausea and diarrhoea reported. Taking with food recommended during training periods. Avoid dairy and calcium-fortified foods at time of dosing.

5 — Recovery-Impact Risks

Tendon and musculoskeletal: Delayed onset tendon symptoms possible months after completing a course. Clinical review warranted at first signs of tendon pain or swelling following recent levofloxacin use.

CNS and sleep: Insomnia and anxiety may affect recovery quality during treatment course.

Microbiome disruption: High. Significant gut microbial diversity reduction reported. Probiotic consideration appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

Iron, calcium, magnesium, zinc, and multivitamins: Significantly reduce levofloxacin absorption. Separate dosing by at least two hours before or six hours after levofloxacin dose.

Dairy and calcium-fortified foods and drinks: Reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Corticosteroids: Concurrent use significantly increases tendon rupture risk. Avoid co-administration where possible. [MHRA 2024]

NSAIDs: Concurrent use may increase risk of CNS side effects including seizures. Caution warranted given prevalence of NSAID use in elite sport.

QTc-prolonging medicines: Additive QTc prolongation risk. Higher QTc signal than ciprofloxacin — greater caution warranted.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £1.19 per 500mg tablet.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Metronidazole
Metronidazole
Nitroimidazole · Tablets (200mg, 400mg) · POM
POM Rx
1 — Athlete-Specific Considerations

Licensed indications include: Bacterial infections caused by anaerobic organisms including dental infections, bacterial vaginosis, and certain gastrointestinal infections. Also used in the treatment and prevention of protozoal infections.

Alcohol interaction: Concurrent alcohol use causes a disulfiram-like reaction: flushing, nausea, vomiting, tachycardia. Avoid alcohol during treatment and for at least 48 hours after completing the course. Highly relevant in team sport environments. See Field 6.

Microbiome impact: Moderate. Primarily disrupts anaerobic flora. Probiotic consideration may be appropriate — see TAF Probiotics entry.

AAD risk: Low to moderate. Lower than broad-spectrum agents but GI side effects common. See Field 4.

Metallic taste: Frequently reported. May affect dietary intake and appetite during treatment course.

2 — Formulation and Route

Form: Tablets (200mg, 400mg). Oral suspension available.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Metronidazole SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Take with or after food to reduce GI side effects. Recommended during training periods to minimise nausea and GI disturbance.

4 — Performance-Impact Risks

GI side effects: Nausea, vomiting, and metallic taste frequently reported. May affect dietary intake, appetite, and training nutrition during treatment course. Taking with food recommended.

AAD risk: Low to moderate. Lower disruption than broad-spectrum agents.

Fatigue and dizziness: Reported with metronidazole use. May affect training tolerance and concentration during treatment course.

Photosensitivity: Not a significant concern. No outdoor training restrictions required.

5 — Recovery-Impact Risks

GI tolerability: Nausea and metallic taste may affect nutrition and hydration targets during treatment course, with downstream impact on recovery.

Microbiome disruption: Moderate. Primarily affects anaerobic flora. Probiotic consideration may be appropriate — see TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

Alcohol: Concurrent use causes a disulfiram-like reaction: flushing, nausea, vomiting, tachycardia. Avoid alcohol during treatment and for at least 48 hours after completing the course. This applies to alcohol in any form including alcohol-containing mouthwashes and some sports recovery products.

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Iron, calcium, magnesium, zinc: No clinically significant absorption interaction established for metronidazole.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.05 per 400mg tablet.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Nitrofurantoin
Nitrofurantoin
Nitrofuran · Capsules (50mg, 100mg MR) · POM
POM Rx
1 — Athlete-Specific Considerations

Licensed indications include: Uncomplicated lower urinary tract infections.

Renal function: Nitrofurantoin requires adequate renal function to achieve therapeutic urinary concentrations. Contraindicated in significant renal impairment. Potential for renal impairment in athletes taking long-term or high-dose NSAIDs worth considering. See SmPC for eGFR thresholds.

Pulmonary toxicity: Rare but serious. Dyspnoea and cough during treatment in an endurance athlete warrants prompt clinical review.

Microbiome impact: Low. Acts locally in the urinary tract with minimal systemic absorption. Lowest microbiome impact of included antibacterials. Probiotic consideration unlikely to be necessary for short courses but may be considered — see TAF Probiotics entry.

AAD risk: Low. Minimal disruption to gut flora compared to systemic antibiotics.

2 — Formulation and Route

Form: Capsules (50mg). Modified-release capsules (100mg). Oral suspension available.

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Nitrofurantoin SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Absorption significantly enhanced when taken with food. Taking with food is recommended and improves bioavailability as well as reducing GI side effects during training.

4 — Performance-Impact Risks

GI side effects: Nausea and vomiting reported, particularly with immediate-release formulations. Modified-release formulation associated with lower GI side effect incidence. Taking with food recommended during training periods.

Pulmonary toxicity: Rare but serious. Dyspnoea and cough during treatment in an endurance athlete warrants prompt clinical review.

AAD risk: Low. Minimal systemic absorption limits gut flora disruption.

Photosensitivity: Not a significant concern. No outdoor training restrictions required.

5 — Recovery-Impact Risks

GI tolerability: Modified-release formulation generally better tolerated than immediate-release. GI side effects unlikely to significantly affect recovery capacity in most athletes on standard short courses.

Microbiome disruption: Low. Minimal systemic absorption means gut flora largely unaffected. Probiotic consideration not routinely required for short courses.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

NSAIDs: No direct pharmacokinetic interaction. However concurrent long-term or high-dose NSAID use may impair renal function, reducing nitrofurantoin efficacy and increasing risk of toxicity. See Field 1.

Antacids containing magnesium trisilicate: Reduce nitrofurantoin absorption and urinary excretion. Avoid concurrent use.

Iron, calcium, magnesium, zinc supplements: No clinically significant absorption interaction established for nitrofurantoin beyond the magnesium trisilicate antacid note above.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.68 per 100mg modified-release capsule.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Trimethoprim
Trimethoprim
Diaminopyrimidine · Tablets (100mg, 200mg) · POM
POM Rx
1 — Athlete-Specific Considerations

Licensed indications include: Urinary tract infections and respiratory tract infections caused by susceptible organisms.

Folate antagonism: Trimethoprim reduces folic acid (folate) availability. In athletes with marginal folate status, including those with restrictive dietary intake or in a RED-S context, this warrants clinical consideration. Also relevant where trimethoprim is prescribed to female athletes who may be or become pregnant.

Microbiome impact: Low. Narrow spectrum limits gut flora disruption.

AAD risk: Low.

Photosensitivity: Mild signal. Relevant for prolonged outdoor training or competition during treatment course. Sun protection advisable.

2 — Formulation and Route

Form: Tablets (100mg, 200mg). Oral suspension available.

Route: Oral

Travel: Tablets — no restrictions. Carry original packaging with dispensing label.

Oral suspensions — check airline carry-on rules for volumes over 100ml. Verify local regulatory status before international travel.

SmPC: Trimethoprim SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Can be taken with or without food. Taking with food recommended to minimise GI side effects during training.

Outdoor training and photosensitivity: Sun protection advisable during prolonged outdoor training or competition during treatment course.

4 — Performance-Impact Risks

GI side effects: Nausea and vomiting reported but generally mild. Taking with food recommended during training periods.

AAD risk: Low. Narrow spectrum limits gut flora disruption and associated diarrhoea risk.

Photosensitivity: Mild signal. Sun protection advisable for outdoor training and competition during treatment course.

Folate availability: Reduced folate availability during treatment course may be relevant in athletes with marginal dietary folate intake.

5 — Recovery-Impact Risks

GI tolerability: Generally well tolerated. GI side effects unlikely to significantly affect recovery capacity in most athletes on standard short courses.

Microbiome disruption: Low. Narrow spectrum means gut flora largely unaffected. Probiotic consideration not routinely required.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive — see SmPC for full interaction profile.

Folate supplements: Athletes taking folate or multivitamins containing folate should be aware that trimethoprim reduces folate availability.

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Iron, calcium, magnesium, zinc: No clinically significant absorption interaction established for trimethoprim.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.27 per 200mg tablet.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Tetracyclines
Class Profiles
Comparative Table
Tetracyclines — Class Overview
Doxycycline · Lymecycline · Minocycline
WADA: Not Prohibited 2026
1 — Athlete-Specific Considerations

Broad-spectrum antibiotics with activity against gram-positive, gram-negative, and atypical organisms.

Licensed indications include: Respiratory tract infections, skin and soft tissue infections, acne vulgaris, Lyme disease, some sexually transmitted infections, and malaria prophylaxis. See individual agent notes for agent-specific licensed indications.

Photosensitivity: Significant class effect. Relevant for all outdoor athletes during treatment course. See Field 3 and individual agent notes.

Supplement and food interactions: Calcium, iron, magnesium, zinc, and dairy products reduce tetracycline absorption via chelation. Separate dosing from these by at least two hours. See Field 6.

Retinoids and high-dose vitamin A: Concurrent use of oral retinoids or vitamin A supplementation above 10,000 IU per day should be avoided. Risk of benign intracranial hypertension. Relevant in athletes using isotretinoin for acne or high-dose vitamin A supplements. [SmPC]

Microbiome impact: Moderate. Varies by agent — see individual agent notes and comparative table.

AAD risk: Moderate. See Field 4.

CNS effects (minocycline): Dizziness, vertigo, and tinnitus reported with minocycline. See individual agent notes.

2 — Formulation and Route

Form: Capsules and tablets (doxycycline, lymecycline, minocycline). Oral suspension available for some formulations.

Route: Oral

Travel: Tablets and capsules — no restrictions. Carry original packaging with dispensing label.

Oral suspensions — check airline carry-on rules for volumes over 100ml. Verify local regulatory status before international travel.

SmPC: See individual agent notes.

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Varies by agent. See individual agent notes. As a general principle, taking with food reduces GI side effects but may reduce absorption for some agents in this class.

Outdoor training and photosensitivity: Avoid prolonged sun exposure during treatment course. Additional sun protection measures required for outdoor training and competition. Wear protective clothing where possible. Photosensitivity risk varies by agent. See individual agent notes.

4 — Performance-Impact Risks

Photosensitivity: Significant class effect. Sunburn, skin reactions, and phototoxicity reported during treatment course. Directly relevant to outdoor training and competition. Sun protection and protective clothing required. Risk varies by agent. See individual agent notes.

GI side effects: Nausea, vomiting, and oesophageal irritation reported across the class. Taking with food and remaining upright after dosing recommended during training periods.

AAD risk: Moderate. GI side effects may affect hydration, electrolyte balance, and training nutrition during treatment course.

CNS effects (minocycline): Dizziness, vertigo, and tinnitus reported. May affect balance, concentration, and training performance. See minocycline individual agent notes.

5 — Recovery-Impact Risks

GI tolerability: GI side effects during a course may affect training nutrition and hydration targets, with downstream impact on recovery capacity.

Microbiome disruption: Moderate. Varies by agent. Probiotic consideration may be appropriate. See TAF Probiotics entry and individual agent notes.

CNS effects (minocycline): Dizziness and vertigo may affect sleep quality and recovery. See minocycline individual agent notes.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive. See individual agent SmPC for full interaction profile.

Calcium, iron, magnesium, zinc, and multivitamins: Reduce tetracycline absorption via chelation. Separation period varies by agent — see individual agent notes.

Dairy and calcium-fortified foods and drinks: Reduce absorption via chelation. Where a meal contains dairy or fortified products, take at least two hours before or six hours after. See individual agent notes for exceptions.

Retinoids and high-dose vitamin A: Concurrent use should be avoided. Risk of benign intracranial hypertension. [SmPC]

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

Oral contraceptives: No clinically significant pharmacokinetic interaction established with tetracyclines based on current evidence. Exception: see minocycline individual agent notes.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Generic oral antibiotics. Low cost through NHS dispensing and private prescription. Indicative costs per unit in individual agent notes.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer and dispensed product. Verify per dispensed product SmPC.

Lactose: Present in some formulations. Verify per dispensed product.

Gelatin: Present in some capsule formulations. Not suitable for vegetarians, vegans, or those observing halal or kosher dietary requirements where gelatin is derived from non-compliant sources. Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

INDIVIDUAL AGENTS

Doxycycline
1st generation tetracycline · Capsules/tablets (50mg, 100mg) · POM
POM Rx
1 — Athlete-Specific Considerations

Licensed indications include: Respiratory tract infections, skin and soft tissue infections, acne vulgaris, Lyme disease, some sexually transmitted infections, and malaria prophylaxis.

Photosensitivity: High risk within this class. Phototoxic reactions reported including severe sunburn and skin blistering. Directly relevant to outdoor athletes. Sun protection and protective clothing essential during treatment course and for a period after stopping.

Microbiome impact: Moderate. Marked short-term decrease in Bifidobacterium diversity reported. A7

AAD risk: Moderate.

Food interaction: Absorption not significantly affected by food or milk per SmPC. Taking with food or milk recommended if gastric irritation occurs.

2 — Formulation and Route

Form: Capsules (50mg, 100mg). Modified-release capsules (40mg, Efracea). Dispersible tablets (100mg, Vibramycin-D).

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Doxycycline SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Absorption not significantly affected by food or milk. Taking with food or milk recommended if gastric irritation occurs. Avoid dairy and calcium-fortified foods at time of dosing where absorption optimisation is a priority.

Administration: Swallow capsules with plenty of water in a sitting or standing position. Take well before retiring at night to reduce the risk of oesophageal irritation and ulceration. [SmPC]

Outdoor training and photosensitivity: Avoid prolonged sun exposure during treatment course and for a period after stopping. Sun protection and protective clothing essential for all outdoor training and competition.

4 — Performance-Impact Risks

Photosensitivity: High risk. Phototoxic reactions including severe sunburn and skin blistering reported. Sun protection and protective clothing essential for outdoor training and competition during treatment course.

GI side effects: Nausea and oesophageal irritation reported. Taking with food and remaining upright after dosing recommended during training periods.

AAD risk: Moderate. GI side effects may affect hydration, electrolyte balance, and training nutrition during treatment course.

5 — Recovery-Impact Risks

GI tolerability: Generally well tolerated when taken with food. GI side effects may affect training nutrition and hydration targets during treatment course.

Microbiome disruption: Moderate. Marked short-term decrease in Bifidobacterium diversity reported. Probiotic consideration may be appropriate. See TAF Probiotics entry. A7

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive. See SmPC for full interaction profile.

Calcium, iron, magnesium, zinc, and multivitamins: Reduce doxycycline absorption via chelation. Separate dosing by at least two hours before or six hours after doxycycline dose.

Dairy and calcium-fortified foods and drinks: Reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Retinoids and high-dose vitamin A: Concurrent use should be avoided. Risk of benign intracranial hypertension. [SmPC]

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.09 per 100mg capsule.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Lymecycline
Tetracycline · Capsules (408mg) · POM
POM Rx
1 — Athlete-Specific Considerations

Licensed indications include: Acne vulgaris and other infections susceptible to tetracycline antibiotics.

Photosensitivity: Moderate risk within this class. Lower photosensitivity signal than doxycycline but still relevant for outdoor athletes. Sun protection advisable during treatment course.

Microbiome impact: Low to moderate. Less well characterised than doxycycline in available evidence.

AAD risk: Low to moderate.

Long-term use: Prolonged use increases cumulative microbiome disruption and photosensitivity exposure risk. Worth noting in athletes on extended courses.

2 — Formulation and Route

Form: Capsules (408mg).

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Lymecycline SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: No specific food guidance in SmPC. Avoid dairy and calcium-fortified foods at time of dosing due to chelation and absorption reduction.

Administration: Swallow capsules with plenty of water in a sitting or standing position. Take well before retiring at night to reduce the risk of oesophageal irritation and ulceration. [SmPC]

Outdoor training and photosensitivity: Avoid prolonged sun exposure during treatment course. Sun protection and protective clothing advisable for outdoor training and competition.

4 — Performance-Impact Risks

Photosensitivity: Moderate risk. Sun protection advisable for outdoor training and competition during treatment course.

GI side effects: Nausea and GI disturbance reported. Ensure adequate fluid intake when dosing. Remaining upright after dosing recommended during training periods.

AAD risk: Low to moderate. GI side effects may affect hydration and training nutrition during treatment course.

Long-term use: Extended courses for acne increase cumulative photosensitivity exposure and microbiome disruption risk.

5 — Recovery-Impact Risks

GI tolerability: Generally well tolerated. GI side effects may affect training nutrition and hydration targets during treatment course.

Microbiome disruption: Low to moderate. Less well characterised than doxycycline. Probiotic consideration may be appropriate for extended courses. See TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive. See SmPC for full interaction profile.

Calcium, iron, magnesium, zinc, and multivitamins: Reduce lymecycline absorption via chelation. Separate dosing by at least two hours before or six hours after lymecycline dose.

Dairy and calcium-fortified foods and drinks: Reduce absorption. Where a meal contains dairy or fortified products, take at least two hours before or six hours after.

Retinoids and high-dose vitamin A: Concurrent use should be avoided. Risk of benign intracranial hypertension. Particularly relevant given lymecycline is commonly co-prescribed with topical retinoids for acne. [SmPC]

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.13 per 408mg capsule.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Minocycline
Tetracycline · Modified-release capsules (100mg) · POM · Minocin MR
POM Rx
1 — Athlete-Specific Considerations

Licensed indications include: Acne vulgaris.

CNS effects: Dizziness commonly reported. Vertigo and tinnitus reported less frequently. May affect balance, coordination, and training performance. Symptoms typically resolve on stopping treatment but warrant clinical review if persistent.

Hyperpigmentation: Reported at various body sites including skin, nails, teeth, and oral mucosa. May develop regardless of dose or duration but more common with long-term use. May persist after stopping treatment. [SmPC]

Photosensitivity: Lower risk than doxycycline within this class. Sun protection still advisable for outdoor athletes.

Microbiome impact: Low to moderate. Less well characterised than doxycycline in available evidence.

AAD risk: Low to moderate.

Long-term use: Prolonged use increases cumulative microbiome disruption risk and is associated with rare but serious adverse effects including drug-induced lupus and hepatotoxicity. Clinical monitoring recommended at three-monthly intervals where treatment exceeds six months. [SmPC]

2 — Formulation and Route

Form: Modified-release capsules (100mg).

Route: Oral

Travel: No restrictions. Carry original packaging with dispensing label. Verify local regulatory status before international travel.

SmPC: Minocycline SmPC ↗

3 — Dose and Timing Around Training

Dosing per SmPC and BNF.

Food: Absorption not significantly impaired by food or moderate amounts of milk. Taking with food recommended to reduce GI side effects during training.

Administration: Swallow capsules with plenty of fluid in a sitting or standing position. Take well before retiring at night to reduce the risk of oesophageal irritation and ulceration. [SmPC]

Supplement timing: Iron, calcium, magnesium, aluminium, bismuth, and zinc salts reduce minocycline absorption. Separate dosing by at least three hours before or after minocycline dose. [SmPC]

Outdoor training and photosensitivity: Photosensitivity risk lower than doxycycline but sun protection still advisable for outdoor training and competition.

4 — Performance-Impact Risks

CNS effects: Dizziness commonly reported. Vertigo and tinnitus reported less frequently. May affect balance, coordination, and training performance during treatment course.

Photosensitivity: Lower risk than doxycycline within this class. Sun protection advisable for outdoor training and competition.

GI side effects: Nausea and GI disturbance reported. Taking with food recommended during training periods.

AAD risk: Low to moderate. GI side effects may affect hydration and training nutrition during treatment course.

Long-term use: Extended courses for acne associated with rare but serious adverse effects. See Field 1.

5 — Recovery-Impact Risks

CNS effects: Dizziness and vertigo may affect sleep quality and recovery during treatment course.

GI tolerability: Generally well tolerated. GI side effects may affect training nutrition and hydration targets during treatment course.

Microbiome disruption: Low to moderate. Probiotic consideration may be appropriate for extended courses. See TAF Probiotics entry.

6 — Medicine and Supplement Interactions

Selected interactions relevant to common athlete use patterns. Not exhaustive. See SmPC for full interaction profile.

Iron, calcium, magnesium, zinc, aluminium, bismuth, and multivitamins: Reduce minocycline absorption. Separate dosing by at least three hours before or after minocycline dose. [SmPC]

Dairy and calcium-fortified foods and drinks: Absorption not significantly impaired by moderate amounts of milk per SmPC. Standard caution applies for calcium-fortified products.

Isotretinoin: Avoid concurrent use and for a period shortly before and after minocycline therapy. Each drug independently associated with benign intracranial hypertension. [SmPC]

Retinoids and high-dose vitamin A: Concurrent use should be avoided. Risk of benign intracranial hypertension. [SmPC]

Oral contraceptives: Minocycline may reduce efficacy of oral contraceptives. [SmPC]

Penicillins: Tetracyclines may interfere with the bactericidal action of penicillins. Avoid concurrent use. [SmPC]

NSAIDs: No direct pharmacokinetic interaction. Concurrent use may compound GI side effects during treatment course.

7 — WADA Status and Anti-Doping Risk Mitigation

WADA: Not Prohibited 2026.

8 — International and Jurisdictional

POM in the UK. Prescription required.

Regulatory and licensing status may vary by jurisdiction. Verify local requirements before international travel or competition.

9 — Club Cost Consideration

Approximately £0.36 per 100mg modified-release capsule.

Verify current pricing at bnf.nice.org.uk.

10 — Allergens, Religious and Lifestyle

Excipients vary by manufacturer. Verify per dispensed product.

Vegetarian: Verify per dispensed product.

Vegan: Verify per dispensed product.

Halal: Verify per dispensed product.

Kosher: Verify per dispensed product.

For product-specific allergen or excipient queries, contact info@medsontrack.com

Further classes in development: Macrolides and Penicillins will be added in subsequent builds.
1Picard M, Robitaille G, Karam F, et al. Cross-reactivity to cephalosporins and carbapenems in penicillin-allergic patients: two systematic reviews and meta-analyses. J Allergy Clin Immunol Pract. 2019;7(8):2722-2738.e5. doi:10.1016/j.jaip.2019.05.038
2Baxter R, Ray GT, Fireman BH. Case-control study of antibiotic use and subsequent Clostridium difficile-associated diarrhea in hospitalized patients. Infect Control Hosp Epidemiol. 2008;29(1):44-50. doi:10.1086/524320
3Nord CE, Heimdahl A, Lundberg C, Marklund G. Impact of cefaclor on the normal human oropharyngeal and intestinal microflora. Scand J Infect Dis. 1987;19(6):681-5. doi:10.3109/00365548709117204
4Gaya H, Adnitt PI, Turner P. Changes in gut flora after cephalexin treatment. BMJ. 1970;3(5723):624-625. doi:10.1136/bmj.3.5723.624
5Vacărean-Trandafir IC, Amărandi RM, Ivanov IC, et al. The impact of cefuroxime prophylaxis on human intestinal microbiota in surgical oncological patients. Front Microbiomes. 2023;1:1092771. doi:10.3389/frmbi.2022.1092771
6Elvers KT, Wilson VJ, Hammond A, et al. Antibiotic-induced changes in the human gut microbiota for the most commonly prescribed antibiotics in primary care in the UK: a systematic review. BMJ Open. 2020;10(9):e035677. doi:10.1136/bmjopen-2019-035677
7Elvers KT, Wilson VJ, Hammond A, et al. Antibiotic-induced changes in the human gut microbiota for the most commonly prescribed antibiotics in primary care in the UK: a systematic review. BMJ Open. 2020;10(9):e035677. doi:10.1136/bmjopen-2019-035677
Cite this entry
Ryan C. Antibacterials. The Athlete's Formulary [Internet]. 2026 [cited 2026 Jul 09]. Available from: theathletesformulary.com/antibacterials